Copper-promoted N-cyclopropylation of anilines and amines by cyclopropylboronic acid.
نویسندگان
چکیده
Reaction of anilines, primary and secondary aliphatic amines with cyclopropylboronic acid in dichloroethane in the presence of Cu(OAc)(2) (1 equiv.), 2,2'-bipyridine (1 equiv.) and sodium carbonate or sodium bicarbonate (2 equiv.) under air atmosphere afforded the corresponding N-cyclopropyl derivatives in good to excellent yields.
منابع مشابه
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ورودعنوان ژورنال:
- Chemical communications
دوره 46 19 شماره
صفحات -
تاریخ انتشار 2010